天然产物 天然产物苯丙素类 Phenylpropanoids
Tetrahydromagnolol (Synonyms: Magnolignan)
Tetrahydromagnolol (Magnolignan)，是 Magnolol 的主要代谢产物，是一种有效的选择性大麻素 CB2 受体激动剂，EC50 为 170 nM，Ki 为 416 nM。Tetrahydromagnolol 对 CB2 受体的选择性比 CB1 受体高 20 倍。Tetrahydromagnolol 也是一种弱的 GPR55 受体拮抗剂。
Tetrahydromagnolol Chemical Structure
CAS No. : 20601-85-8
| 规格 | 价格 | 是否有货 | |
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| 1 mg | ￥700 | 询问价格 & 货期 | |
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| 生物活性 |
Tetrahydromagnolol (Magnolignan), a main metabolite of Magnolol, is a potent and selective cannabinoid CB2 receptor agonist with an EC50 of 170 nM and a Ki of 416 nM. Tetrahydromagnolol possesses 20-fold more selective for CB2 receptor than CB1 receptor. Tetrahydromagnolol is also a weak GPR55 receptor antagonist[1]. |
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| IC50 & Target[1] |
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| 分子量 |
270.37 |
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| Formula |
C18H22O2 |
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| CAS 号 |
20601-85-8 |
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| 中文名称 |
四氢厚朴酚 |
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| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
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| 储存方式 |
Please store the product under the recommended conditions in the Certificate of Analysis. |
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| 参考文献 |
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