PG106;
PG106 是一种有效的、选择性的 hMC3 receptor 拮抗剂 (IC50= 210 nM)，对 hMC4 受体(EC50=9900 nM) 和 hMC5 受体无活性。
PG106 Chemical Structure
CAS No. : 944111-22-2
| 规格 | 是否有货 | ||
|---|---|---|---|
| 100 mg | ; | 询价 | ; |
| 250 mg | ; | 询价 | ; |
| 500 mg | ; | 询价 | ; |
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PG106 的其他形式现货产品:
| 生物活性 |
PG106 is a potent and selective human melanocortin 3 (hMC3) receptor antagonist (IC50=210 nM) and has noactivity at hMC4 receptors (EC50=9900 nM) and hMC5 receptor[1]. |
IC50 Target |
IC50: 210 nM (hMC3 receptor)EC50: 9900 nM (hMC4 receptor)[1] |
|---|---|
| 分子量 |
1008.18 |
| Formula |
C51H69N13O9 |
| CAS 号 |
944111-22-2 |
| Sequence Shortening |
Ac-{Nle}-D-{Bal}-{D-Nal}-RWK-NH2 (Lactam bridge:Asp2-Lys7) |
| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
| 储存方式 |
Please store the product under the recommended conditions in the Certificate of Analysis. |
| 参考文献 |
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