天然产物 天然产物苯丙素类 Phenylpropanoids
Coniferyl ferulate (Synonyms: 阿魏酸松柏酯) 纯度: 98.56%
Coniferyl ferulate 是一种强效的谷胱甘肽 S-转移酶 (GST) 抑制剂,可逆转多药耐药性并下调 P-糖蛋白。Coniferyl ferulate 强抑制人胎盘型谷胱甘肽 S-转移酶,IC50 为 0.3 μM。
Coniferyl ferulate Chemical Structure
CAS No. : 63644-62-2
规格 | 价格 | 是否有货 | 数量 |
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1 mg | ¥1000 | In-stock | |
5 mg | ¥2500 | In-stock | |
10 mg | ¥4200 | In-stock | |
50 mg | 询价 | ||
100 mg | 询价 |
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Coniferyl ferulate 相关产品
•相关化合物库:
- Natural Product Library Plus
- Bioactive Compound Library Plus
- Membrane Transporter/Ion Channel Compound Library
- Metabolism/Protease Compound Library
- Natural Product Library
- Anti-Cancer Compound Library
- Antioxidants Compound Library
- Oxygen Sensing Compound Library
- Phenols Library
- Traditional Chinese Medicine Monomer Library
生物活性 |
Coniferyl ferulate, a strong inhibitor of glutathione S-transferase (GST), reverses multidrug resistance and downregulates P-glycoprotein. Coniferyl ferulate shows strong inhibition of human placental GST with an IC50 of 0.3 μM[1]. |
IC50 & Target |
Glutathione S-transferase[1] |
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分子量 |
356.37 |
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Formula |
C20H20O6 |
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CAS 号 |
63644-62-2 |
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中文名称 |
阿魏酸松柏酯 |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
4°C, protect from light *In solvent : -80°C, 6 months; -20°C, 1 month (protect from light) |
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溶解性数据 |
In Vitro:
DMSO : 100 mg/mL (280.61 mM; Need ultrasonic) 配制储备液
*
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 In Vivo:
请根据您的实验动物和给药方式选择适当的溶解方案。以下溶解方案都请先按照 In Vitro 方式配制澄清的储备液,再依次添加助溶剂: ——为保证实验结果的可靠性,澄清的储备液可以根据储存条件,适当保存;体内实验的工作液,建议您现用现配,当天使用; 以下溶剂前显示的百
*以上所有助溶剂都可在 MCE 网站选购。
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参考文献 |
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