天然产物 天然产物苯丙素类 Phenylpropanoids
8-Geranyloxypsoralen (Synonyms: 8-香叶草氧基补骨脂素) 纯度: 99.93%
8-Geranyloxypsoralen 是从葡萄柚中分离出的一种呋喃香豆素,能作为 P450 3A4 (CYP3A4) 的有效抑制剂,其 IC50 值为 3.93 μM。
8-Geranyloxypsoralen Chemical Structure
CAS No. : 7437-55-0
规格 | 价格 | 是否有货 | 数量 |
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5 mg | ¥4030 | In-stock | |
10 mg | ¥6860 | In-stock | |
50 mg | 询价 | ||
100 mg | 询价 |
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8-Geranyloxypsoralen 相关产品
•相关化合物库:
- Natural Product Library Plus
- Bioactive Compound Library Plus
- Metabolism/Protease Compound Library
- Natural Product Library
- Anti-Cancer Compound Library
- Anti-Aging Compound Library
- Antioxidants Compound Library
- Oxygen Sensing Compound Library
- Food-Sourced Compound Library
- Targeted Diversity Library
生物活性 |
8-Geranyloxypsoralen is a furanocoumarin isolated from grapefruit, acts as a potent inhibitor of P450 3A4 (CYP3A4) with an IC50 of 3.93 μM[1]. |
IC50 & Target |
IC50: 3.93 μM (P450 3A4)[1] |
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分子量 |
338.40 |
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Formula |
C21H22O4 |
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CAS 号 |
7437-55-0 |
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中文名称 |
8-香叶草氧基补骨脂素 |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
4°C, protect from light *In solvent : -80°C, 6 months; -20°C, 1 month (protect from light) |
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溶解性数据 |
In Vitro:
DMSO : 100 mg/mL (295.51 mM; Need ultrasonic) 配制储备液
*
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 In Vivo:
请根据您的实验动物和给药方式选择适当的溶解方案。以下溶解方案都请先按照 In Vitro 方式配制澄清的储备液,再依次添加助溶剂: ——为保证实验结果的可靠性,澄清的储备液可以根据储存条件,适当保存;体内实验的工作液,建议您现用现配,当天使用; 以下溶剂前显示的百
*以上所有助溶剂都可在 MCE 网站选购。
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参考文献 |
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