DAMGO (TFA)

发表于由

DAMGO (TFA); 纯度: 99.76%

DAMGO TFA 是一种选择性的 μ-阿片受体 (μ-OPR) 激动剂，Kd 值为 3.46 nM。

DAMGO (TFA)amp;;

DAMGO (TFA) Chemical Structure

CAS No. : 950492-85-0

规格 价格 是否有货 数量
10;mM;*;1 mL in Water ￥1367 In-stock
1 mg ￥600 In-stock
5 mg ￥990 In-stock
10 mg ￥1700 In-stock
25 mg ￥3700 In-stock
50 mg ; 询价 ;
100 mg ; 询价 ;

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DAMGO (TFA) 相关产品

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生物活性

DAMGO TFA is a μ-opioid receptor (μ-OPR ) selective agonist with a Kd of 3.46 nM for native μ-OPR[1].

分子量

627.61

Formula

C28H36F3N5O8
CAS 号

950492-85-0
Sequence

Tyr-{d-Ala}-Gly-{Me-Phe}-Gly-ol
Sequence Shortening

Y-{d-Ala}-G-{Me-Phe}-G-ol
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Sealed storage, away from moisture

Powder -80deg;C 2 years
-20deg;C 1 year

*In solvent : -80deg;C, 6 months; -20deg;C, 1 month (sealed storage, away from moisture)
溶解性数据
In Vitro:;

H2O : 125 mg/mL (199.17 mM; Need ultrasonic)

配制储备液
浓度 溶剂体积 质量 1 mg 5 mg 10 mg
1 mM 1.5933 mL 7.9667 mL 15.9335 mL
5 mM 0.3187 mL 1.5933 mL 3.1867 mL
10 mM 0.1593 mL 0.7967 mL 1.5933 mL

*

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)。-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
参考文献

  • [1]. FEBS Lett. 1995 Jan 2;357(1):93-7. Onogi T, et al. DAMGO, a mu-opioid receptor selective agonist, distinguishes between mu- and delta-opioid receptors around their first extracellular loops.