HS024 TFA; 纯度: 99.63%
HS024 是一种选择性的 MC4 受体拮抗剂,对 MC4、MC5、MC3 和 MC1 的 Ki 分别为 0.29、3.29、5.45 和 18.6 nM。HS024 增加食物摄入。
HS024 TFA Chemical Structure
规格 | 价格 | 是否有货 | 数量 |
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1 mg | ¥1400 | In-stock | |
5 mg | ¥3200 | In-stock | |
10 mg | ¥5200 | In-stock | |
50 mg | ; | 询价 | ; |
100 mg | ; | 询价 | ; |
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HS024 TFA 相关产品
bull;相关化合物库:
- Bioactive Compound Library Plus
- GPCR/G Protein Compound Library
- Neuronal Signaling Compound Library
- Peptide Library
生物活性 |
HS024 is a selective MC4 receptor antagonist, with Kis of 0.29, 3.29, 5.45, 18.6 nM for MC4, MC5, MC3, and MC1, respectively. HS024 increase food intake[1]. |
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分子量 |
1380.52 |
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Formula |
C60H80F3N19O12S2 |
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Sequence Shortening |
Ac-C-{Nle}-RH-{D-2Nal}-RWGC-NH2 (Disulfide bridge:Cys1-Cys9) |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
Sealed storage, away from moisture
*In solvent : -80deg;C, 6 months; -20deg;C, 1 month (sealed storage, away from moisture) |
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溶解性数据 |
In Vitro:;
H2O : 50 mg/mL (36.22 mM; Need ultrasonic) 配制储备液
*
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |
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参考文献 |
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