HS024

发表于由

HS024;

HS024 是一种选择性的 MC4 受体拮抗剂，对 MC4、MC5、MC3 和 MC1 的 Ki 分别为 0.29、3.29、5.45 和 18.6 nM。HS024 增加食物摄入。

HS024amp;;

HS024 Chemical Structure

CAS No. : 212370-59-7

规格 是否有货
5 mg 询价
10 mg 询价

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生物活性

HS024 is a selective MC4 receptor antagonist, with Kis of 0.29, 3.29, 5.45, and 18.6 nM for MC4, MC5, MC3, and MC1, respectively. HS024 increase food intake[1].

分子量

1266.50

Formula

C58H79N19O10S2
CAS 号

212370-59-7
Sequence Shortening

Ac-C-{Nle}-RH-{D-2Nal}-RWGC-NH2 (Disulfide bridge:Cys1-Cys9)
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Kask A, et al. Discovery of a novel superpotent and selective melanocortin-4 receptor antagonist (HS024): evaluation in vitro and in vivo. Endocrinology. 1998;139(12):5006-5014.