G-Protein antagonist peptide

发表于由

G-Protein antagonist peptide;

G-Protein antagonist peptide 是一种 substance P 相关肽，可抑制 G 蛋白与其受体的结合。G-Protein antagonist peptide 竞争性和可逆性地抑制毒蕈碱型乙酰胆碱受体 M2 (M2 muscarinic receptor) 对 Gi 或 Go 的激活，并通过 β-肾上腺素受体抑制 Gs 的激活。

G-Protein antagonist peptideamp;;

G-Protein antagonist peptide Chemical Structure

CAS No. : 143675-79-0

规格 是否有货
100 mg ; 询价 ;
250 mg ; 询价 ;
500 mg ; 询价 ;

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生物活性

G-Protein antagonist peptide is the substance P-related peptide that inhibits binding of G proteins to their receptors. G-Protein antagonist peptide competitively and reversibly inhibits M2 muscarinic receptor activation of Gi or Go and inhibits Gs activation by β-adrenoceptors.

分子量

1093.26

Formula

C5H7FN2O2W3
CAS 号

143675-79-0
Sequence

{Glp}-Gln-Trp-Phe-Trp-Trp-Met-NH2
Sequence Shortening

{Glp}QWFWWM-NH2
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Mukai H, et al. G protein antagonists. A novel hydrophobic peptide competes with receptor for G protein binding. J Biol Chem. 1992;267(23):16237-16243.